Lukáš Tenora: search on Z-Library

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1

N -(Pivaloyloxy)alkoxy-carbonyl Prodrugs of the Glutamine Antagonist 6-Diazo-5-oxo-L-norleucine (DON) as a Potential Treatment for HIV Associated Neurocognitive Disorders

Nedelcovych, Michael T., Tenora, Lukáš, Kim, Boe-Hyun, Kelschenbach, Jennifer, Chao, Wei, Hadas, Eran, Jančařík, Andrej, Prchalová, Eva, Zimmermann, Sarah C., Dash, Ranjeet P., Gadiano, Alexandra J.,

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 712 KB

english, 2017

2

Discovery of 6-Diazo-5-oxo-L-norleucine (DON) prodrugs with enhanced CSF delivery in monkeys: a potential treatment for glioblastoma

Rais, Rana, Jancarik, Andrej, Tenora, Lukas, Nedelcovych, Michael, Alt, Jesse, Englert, Judson, Rojas, Camilo, Le, Anne, Elgogary, Amira, Tan, Jessica, Monincova, Lenka, Pate, Kelly, Adams, Robert J.,

Journal:

Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 688 KB

english, 2016

3

N-substituted prodrugs of mebendazole provide improved aqueous solubility and oral bioavailability in mice and dogs

Zimmermann, Sarah C., Tichy, Tomas, Vavra, Jan, Dash, Ranjeet P., Slusher, C. Ethan, Gadiano, Alexandra J, Wu, Ying, Jančařík, Andrej, Tenora, Lukáš, Monincova, Lenka, Prchalova, Eva, Riggins, Gregory

Journal:

Journal of Medicinal Chemistry

Year:

2018

Language:

english

File:

PDF, 558 KB

english, 2018

4

Enhanced Brain Delivery of (2-(phosphonomethyl)pentanedioic acid) following Intranasal Administration of its γ-substituted Ester Prodrugs

Nedelcovych, Michael, Dash, Ranjeet P., Tenora, Lukáš, Zimmermann, Sarah C., Gadiano, Alexandra J, Garrett, Caroline, Alt, Jesse, Hollinger, Kristen R., Pommier, Elie, Jančařík, Andrej, Rojas, Camilo,

Journal:

Molecular Pharmaceutics

Year:

2017

Language:

english

File:

PDF, 616 KB

english, 2017

5

A new and facile synthesis of methyl 3-amino-4,5,6,7-tetrahydrobenzo[b]thiophene-2-carboxylate

Lukáš Tenora, Marian Buchlovič, Stanislav Man, Milan Potáček

Journal:

Tetrahedron Letters

Year:

2011

Language:

english

File:

PDF, 307 KB

english, 2011

6

Application of Pd-Catalyzed Cross-Coupling Reactions in the Synthesis of 5,5-Dimethyl-5,6-dihydro-4-Η-pyrrolo[1,2-b]pyrazoles that inhibit ALK5 Kinase

Tenora, Lukas, Galeta, Juraj, Řezníčková, Eva, Krystof, Vladimir, Potacek, Milan

Journal:

Journal of Organic Chemistry

Year:

2016

Language:

english

File:

PDF, 1.39 MB

english, 2016

7

Discovery of a para-acetoxy-benzyl ester prodrug of a hydroxamate-based Glutamate Carboxypeptidase II inhibitor as oral therapy for neuropathic pain

Rais, Rana, Vávra, Jan, Tichý, Tomáš, Dash, Ranjeet P., Gadiano, Alexandra J., Tenora, Lukas, Monincova, Lenka, Barinka, Cyril, Alt, Jesse, Zimmermann, Sarah C., Slusher, C. Ethan, Wu, Ying, Wozniak,

Journal:

Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 555 KB

english, 2017

8

Identification of Novel Carbonic Anhydrase IX Inhibitors Using High-Throughput Screening of Pooled Compound Libraries by DNA-Linked Inhibitor Antibody Assay (DIANA)

Tykvart, Jan, NavrÃ¡til, VÃ¡clav, Kugler, Michael, Å Ã¡cha, Pavel, Schimer, JiÅÃ, HlavÃ¡ÄkovÃ¡, Anna, Tenora, LukÃ¡Å¡, ZemanovÃ¡, Jitka, Dejmek, Milan, KrÃ¡l, Vlastimil, PotÃ¡Äek, Milan, Majer, Pa

Journal:

Year:

2020

File:

PDF, 770 KB

2020

9

Enhanced oral bioavailability of 2-(phosphonomethyl)-pentanedioic acid (2-PMPA) from its (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl (ODOL) based prodrugs

Dash, Ranjeet P., Tichý, Tomáš, Veeravalli, Vijayabhaskar, Lam, Jenny, Alt, Jesse, Wu, Ying, Tenora, Lukáš, Majer, Pavel, Slusher, Barbara S., Rais, Rana

Journal:

Molecular Pharmaceutics

Year:

2019

File:

PDF, 421 KB

2019

10

Discovery of Orally Available Prodrugs of the Glutamate Carboxypeptidase II (GCPII) Inhibitor 2-Phosphonomethylpentanedioic Acid (2-PMPA)

Majer, Pavel, Jančařík, Andrej, Krečmerová, Marcela, Tichý, Tomáš, Tenora, Lukáš, Wozniak, Krystyna, Wu, Ying, Pommier, Elie, Ferraris, Dana, Rais, Rana, Slusher, Barbara S.

Journal:

Journal of Medicinal Chemistry

Year:

2016

Language:

english

File:

PDF, 495 KB

english, 2016

11

1,3-Dipolar Cycloaddition in the Preparation of New Fused Heterocyclic Compounds via Thermal Initiation

Porubský, Martin, Tenora, Lukáš, Potáček, Milan

Journal:

Year:

2016

Language:

english

File:

PDF, 2.19 MB

english, 2016

12

ALK5 kinase inhibitory activity and synthesis of 2,3,4-substituted 5,5-dimethyl-5,6-dihydro-4 H -pyrrolo[1,2- b ]pyrazoles

Řezníčková, Eva, Tenora, Lukáš, Pospíšilová, Pavlína, Galeta, Juraj, Jorda, Radek, Berka, Karel, Majer, Pavel, Potáček, Milan, Kryštof, Vladimír

Journal:

European Journal of Medicinal Chemistry

Year:

2017

Language:

english

File:

PDF, 1.22 MB

english, 2017

13

Tumor-targeted delivery of 6-Diazo-5-oxo-L-norleucine (DON) using substituted acetylated lysine prodrugs

Tenora, Lukáš, Alt, Jesse, Dash, Ranjeet P., Gadiano, Alexandra J, Novotna, Katerina, Veeravalli, Vijayabhaskar, Lam, Jenny, Kirkpatrick, Quinn R, Lemberg, Kathryn, Majer, Pavel, Rais, Rana, Slusher,

Journal:

Journal of Medicinal Chemistry

Year:

2019

Language:

english

File:

PDF, 606 KB

english, 2019

14

Tumor-targeted delivery of 6-Diazo-5-oxo-L-norleucine (DON) using substituted acetylated lysine prodrugs

Tenora, Lukáš, Alt, Jesse, Dash, Ranjeet P., Gadiano, Alexandra J, Novotna, Katerina, Veeravalli, Vijayabhaskar, Lam, Jenny, Kirkpatrick, Quinn R, Lemberg, Kathryn, Majer, Pavel, Rais, Rana, Slusher,

Journal:

Journal of Medicinal Chemistry

Year:

2019

File:

PDF, 606 KB

2019

15

Dihydropyrrolo[1,2-b]pyrazoles: withasomnine and related compounds

Galeta, Juraj, Tenora, Lukáš, Man, Stanislav, Potáček, Milan

Journal:

Year:

2013

Language:

english

File:

PDF, 10.35 MB

english, 2013

16

Enhanced oral bioavailability of 2-(phosphonomethyl)-pentanedioic acid (2-PMPA) from its (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl (ODOL) based prodrugs

Dash, Ranjeet P., Tichý, Tomáš, Veeravalli, Vijayabhaskar, Lam, Jenny, Alt, Jesse, Wu, Ying, Tenora, Lukáš, Majer, Pavel, Slusher, Barbara S., Rais, Rana

Journal:

Molecular Pharmaceutics

Year:

2019

Language:

english

File:

PDF, 421 KB

english, 2019

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